Peptide Active Data Details
Basic Peptide Information
DICL ID
DICL_Pep_04589
Ion Channel
Intermediate conductance calcium-activated potassium channel protein 4
Peptide Function
Blocker
Gene Name
KCNN4
Activity Data (nM)
IC50
3300 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified
Sequence Information
Peptide Sequence
XFTNVSCTTSKECWSVCQRLHNTSRGKCMNKKCRCYS
Peptide UniProt Accession
UniParc
Not available
Peptide Synonyms/Alias
[CHARYBDOTOXIN; Lqh alpha IT Recombinant; 95751-30-7; 115422-61-2; CTX Toxin; CHARYBDOTOXIN (Native); ChTX; Quinquestriatus Toxin; Charybdotoxin (reduced)]
Peptide Species
Leiurus hebraeus (Hebrew deathstalker scorpion) (Leiurus quinquestriatus hebraeus)
Peptide Name
Potassium channel toxin alpha-KTx 1.1
CAS Number
95751-30-7
Experimental Conditions
pH
pH 7.4
Holding Potential (mV)
Not specified
Temperature
37 °C
Test Method
Efflux Assay (86Rb+)
Test Species
Rattus norvegicus glioma cells
Binding Information
Binding Site
Not specified
Binding Site Residue
Not specified
Ion Channel Information
Gene Abbreviation (ABB)
KCa
Ion Channel UniProt Accession
Source Organism
Rattus norvegicus (Rat)
References & Disease Information
Disease
Not specified
PubChem CID
URL
Not available
PMID
Patent
Not available